Overall Score3.5
- Generality
- Reagent Availability
- Experimental User Friendliness
- Criteria #4
- Criteria #5
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General Characteristics
2-Oxygenated indoles can be synthesized from the corresponding secondary aryl amines and bisulfite adduct of glyoxal.
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General References
- Hinsberg, O. Ber. Dtsch. Chem. Ges. 1888, 21, 110; 1898, 31, 250; 1908, 41, 1367.
- Hinsberg, O.; Rosenzweig, J. Ber. Dtsch. Chem. Ges. 1894, 27, 3253
- Burton, H. J. Chem. Soc. 1932, 546.
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Reaction Mechanism
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Examples
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Experimental Procedure
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Experimental Tips
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References
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Related Reactions
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Related Books
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External Links